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An orexin receptors agonist. It can stimulate feeding following central administration. Synonyms: Human orexin B (TFA); Arg-Ser-Gly-Pro-Pro-Gly-Leu-Gln-Gly-Arg-Leu-Gln-Arg-Leu-Leu-Gln-Ala-Ser-Gly-Asn-His-Ala-Ala-Gly-Ile-Leu-Thr-Met-NH2.TFA; L-arginyl-L-seryl-glycyl-L-prolyl-L-prolyl-glycyl-L-leucyl-L-glutaminyl-glycyl-L-arginyl-L-leucyl-L-glutaminyl-L-arginyl-L-leucyl-L-leucyl-L-glutaminyl-L-alanyl-L-seryl-glycyl-L-asparagyl-L-histidyl-L-alanyl-L-alanyl-glycyl-L-isoleucyl-L-leucyl-L-threonyl-L-methioninamide trifluoroacetic acid. Grade: ≥98%. Molecular formula: C123H212N44O35S.C2HF3O2. Mole weight: 3013.36.
Orexin B (rat, mouse)
An orexin receptors agonist. It can stimulate feeding following central administration. Synonyms: Rat orexin B; Orexin B (mouse); H-Arg-Pro-Gly-Pro-Pro-Gly-Leu-Gln-Gly-Arg-Leu-Gln-Arg-Leu-Leu-Gln-Ala-Asn-Gly-Asn-His-Ala-Ala-Gly-Ile-Leu-Thr-Met-NH2; L-arginyl-L-prolyl-glycyl-L-prolyl-L-prolyl-glycyl-L-leucyl-L-glutaminyl-glycyl-L-arginyl-L-leucyl-L-glutaminyl-L-arginyl-L-leucyl-L-leucyl-L-glutaminyl-L-alanyl-L-asparagyl-glycyl-L-asparagyl-L-histidyl-L-alanyl-L-alanyl-glycyl-L-isoleucyl-L-leucyl-L-threonyl-L-methioninamide. Grade: ≥95% by HPLC. CAS No. 202801-92-1. Molecular formula: C126H215N45O34S. Mole weight: 2936.39.
Orexin B, rat, mouse
Orexin B, rat, mouse (Rat orexin B) is an endogenous agonist at Orexin receptor with K i s of 420 and 36 nM for OX1 and OX2, respectively. Uses: Scientific research. Group: Peptides. Alternative Names: Rat orexin B; Orexin B (mouse). CAS No. 202801-92-1. Pack Sizes: 1 mg; 5 mg; 10 mg. Product ID: HY-P1349.
Orexin receptor antagonist 2
Orexin receptor antagonist 2 (compound 30) is a potent orexin receptor antagonist with pK i s of 7.69 and 9.78. Orexin receptor antagonist 2 has the potential for the research of insomnia [1]. Uses: Scientific research. Group: Signaling pathways. CAS No. 1457940-75-8. Pack Sizes: 10 mM * 1 mL; 5 mg; 10 mg; 25 mg; 50 mg. Product ID: HY-136922.
Orexin receptor antagonist 3
Orexin receptor antagonist 3 (example 216) is an orexin receptor antagonist, which is extracted from the patent WO2011050198A1 [1]. Uses: Scientific research. Group: Signaling pathways. CAS No. 1293282-55-9. Pack Sizes: 10 mM * 1 mL; 5 mg; 10 mg; 25 mg; 50 mg. Product ID: HY-137093.
Orfamide A
It is the major component of a family of cyclic lipopeptides produced by pseudomonas fluorescens pf-5. It is a moderate antifungal agent. It has a profound effect on the swarming motility of bacteria on agar surfaces. Synonyms: N-(3-hydroxy-1-oxotetradecyl)-L-leucyl-D-α-glutamyl-D-allothreonyl-D-alloisoleucyl-L-leucyl-D-seryl-L-leucyl-L-leucyl-D-seryl-L-valine, (10→3)-lactone. Grade: >98% by HPLC. CAS No. 939960-34-6. Molecular formula: C64H114N10O17. Mole weight: 1295.65.
Orfamide B
It is a component of a family of cyclic lipopeptides produced by pseudomonas fluorescens pf-5. Synonyms: N-(3-hydroxy-1-oxotetradecyl)-L-leucyl-D-α-glutamyl-D-allothreonyl-D-valyl-L-leucyl-D-seryl-L-leucyl-L-leucyl-D-seryl-L-valine, (10→3)-lactone. Grade: >98% by HPLC. CAS No. 939960-35-7. Molecular formula: C63H112N10O17. Mole weight: 1281.62.
Orforglipron
Orforglipron (LY3502970) (Compound 67) is an orally active agonist for Glucagon-like peptide-1 receptor ( GLP-1R ), which exhibits potency in ameliorates the type 2 diabete [1]. Uses: Scientific research. Group: Signaling pathways. Alternative Names: LY3502970; GLP-1 receptor agonist 1. CAS No. 2212020-52-3. Pack Sizes: 10 mM * 1 mL; 5 mg; 10 mg; 25 mg. Product ID: HY-112185.
Orforglipron hemicalcium hydrate
Orforglipron hemicalcium hydrate (LY3502970 hemicalcium hydrate; GLP-1 receptor agonist 1 hemicalcium hydrate) is the calcium salt hydrate form of Orforglipron (HY-112185). Orforglipron is an orally active agonist for Glucagon-like peptide-1 receptor (GLP-1R), which exhibits potency in ameliorating the type 2 diabete[1]. Uses: Scientific research. Group: Signaling pathways. Alternative Names: LY3502970 hemicalcium hydrate; GLP-1 receptor agonist 1 hemicalcium hydrate. CAS No. 3008544-96-2. Pack Sizes: 10 mM * 1 mL; 5 mg; 10 mg; 25 mg; 50 mg; 100 mg. Product ID: HY-112185A.
Org 12962 hydrochloride
Org 12962 hydrochloride. Group: Biochemicals. Grades: Purified. CAS No. 210821-63-9. Pack Sizes: 10mg, 50mg. US Biological Life Sciences.
Worldwide
Org 20599
Hoechst 33342 is a cell-permeable fluorescent DNA stain. It binds minor groove of AT-rich regions and is used to quantify DNA in viable cells. Group: Biochemicals. Grades: Highly Purified. CAS No. 156685-94-8. Pack Sizes: 10mg, 50mg. Molecular Formula: C25H40ClNO3, Molecular Weight: 438.04. US Biological Life Sciences.
Worldwide
Org 24598 lithium salt
Org 24598 lithium salt. Group: Biochemicals. Grades: Purified. CAS No. 722456-08-8. Pack Sizes: 10mg, 50mg. US Biological Life Sciences.
Worldwide
Org 25543 hydrochloride
Org 25543 hydrochloride. Group: Biochemicals. Grades: Purified. CAS No. 495076-64-7. Pack Sizes: 10mg, 50mg. US Biological Life Sciences.
Worldwide
Org 25543 hydrochloride
Org 25543 hydrochloride is a selective and irreversible GlyT2 inhibitor ( IC 50 : 16 nM). Org 25543 hydrochloride has analgesia effect. Org 25543 hydrochloride ameliorates mechanical allodynia after partial sciatic nerve ligation injury in mice [1] [2] [3]. Uses: Scientific research. Group: Signaling pathways. CAS No. 495076-64-7. Pack Sizes: 5 mg. Product ID: HY-107527.
Org-26576
Org-26576 is a positive allosteric modulator of AMPA receptor. Org-26576 increases the anteroventral and laterodorsal thalamus, cingulate cortex, dentate gyrus and CA3 subfield of the hippocampus in mice. Org-26576 is potentially used for the treatment of depression and attention deficit disorder. Uses: Potential treatment of depression and attention deficit disorder. Synonyms: Org26576; Org 26576. CAS No. 1026791-61-6. Molecular formula: C11H12N2O2. Mole weight: 204.229.